Nā ʻike huahana
ʻO ka dihydroartemisinin he mea ia o artemisinin, nona ka hopena pepehi ikaika a me ka wikiwiki i ka pae erythrocytic o nā maʻi malaria, a hiki ke hoʻomalu koke i nā hōʻeha a me nā hōʻailona.
1, mea kanu kumu
ʻO ka dihydroartemisinin kahi derivative artemisinin.ʻO Artemisinin kahi lāʻau antimalarial i lawe ʻia mai Artemisia annua.
2、 Hana
Ua like ka hana pharmacological o dihydroartemisinin me ka artemisinin.ʻO ka hopena o ka artemisinin ma ka ultrastructure o Plasmodium falciparum i ka pae erythrocytic ka mea nui e hoʻololi i kona ʻano membrane.Hana mua ka lāʻau lapaʻau i ka membrane vesicle meaʻai, membrane surface a me mitochondria, a ukali ʻia e ka membrane nuklea a me ka endoplasmic reticulum.Eia kekahi, pili ia i ka chromatin i loko o ka nucleus.Hiki iā ia ke hana ma luna o ka membrane vesicle meaʻai, kaohi ʻana i ka pae mua loa o ka ʻai ʻana i ka meaʻai o ka malaria parasite, ka mea e pōloli koke ai ka malaria parasite i nā waikawa amino, hana koke i nā vesicle autophagic, a hoʻokuʻu mau i waho o ke kino, nalowale ka nui cytoplasm a me nā meaʻai, akā ʻaʻole i hoʻohui ʻia, no laila make koke ia.ʻO kāna ʻano hana ka mea nui e hoʻopilikia i ka hana o Plasmodium surface membrane mitochondria.Ma o kona alahaka peroxide (dioxygen) i loko, ua hoʻopili ʻia e ka hao manuahi i hana ʻia ma hope o ka decomposition o ka hemoglobin e hana i nā radical manuahi manuahi a me / a i ʻole nā mea waena electrophilic, a laila hana i nā covalent addducts me nā protein o ka malaria parasite, ka hopena. ka make ana o ka ma'i malaria.ʻO ka lawe ʻia ʻana o ka tritium i kapa ʻia ʻo isoleucine e Plasmodium falciparum moʻomeheu i loko o ka vitro i hōʻike pū ʻia ʻo kāna ʻano hana mua paha ke kāohi i ka synthesis o ka protein Plasmodium.
3、 kahua noi
1. ʻOihana lāʻau lapaʻau
Nā Kūlana Huahana
KULA HANA | |
inoa mea kūʻai | ʻO ka dihydroartemisinin |
CAS | 81496-82-4 |
ʻO ke kimekema | C15H24O5 |
Brand | Hʻo ʻaneʻi |
Mmea hana | Yunnan Hande Bio-Tech Co., Ltd. |
Cʻāina | Kunming,China |
Hoʻokumu ʻia | 1993 |
BʻIkepili ASIC | |
Nā huaʻōlelo like | (3R,5aS,6R,8aS,9R,12S,12aR)-octahydrogen -3,6,9-trimethyl -3,12-epoxy -12H-pyrane [4,3-j]-1,2-coumaron -10 (3H) waiʻona;Dihydroartemisinin;Dihxdroarteannui;Dihydroartemisinin USP/EP/BP |
Kapili | |
Kaumaha | 284.35 |
HS Code | N/A |
ʻAno maikaʻiShoʻopaʻapaʻa | Hōʻikeʻike Hui |
Cpalapala hōʻoia | N/A |
Hoʻāʻo | Hoʻopilikino ʻia e like me nā pono o ka mea kūʻai aku |
Ka nana aku | He aniani keʻokeʻo |
ʻano o ka unuhi ʻana | Artemisia annua Linn. |
Makahiki Makahiki | Hoʻopilikino ʻia e like me nā pono o ka mea kūʻai aku |
Pūʻolo | Hoʻopilikino ʻia e like me nā pono o ka mea kūʻai aku |
Hana Hoao | HPLC |
Loko | lehulehuhalihalis |
PhāʻawiTerms | T/T, D/P, D/A |
Other | E ʻae i ka loiloi mea kūʻai aku i nā manawa a pau;E kōkua i nā mea kūʻai aku me ka hoʻopaʻa inoa hoʻoponopono. |
Hōʻike huahana Hande
1. ʻO nā huahana a pau i kūʻai ʻia e ka ʻoihana he semi-finished maka.Kuhi nui ʻia nā huahana i nā mea hana me nā hōʻailona hana, a ʻaʻole nā mea waiwai nā huahana hope loa.
2. ʻO ka pono kūpono a me nā noi i komo i ka hoʻolauna mai nā palapala i paʻi ʻia.ʻAʻole ʻōlelo ka poʻe i ka hoʻohana pololei ʻana, a hōʻole ʻia nā kūʻai kūʻai.
3. ʻO nā kiʻi a me nā ʻike huahana ma kēia pūnaewele no ka kuhikuhi wale nō, a e lanakila ka huahana maoli.